Aspadol 100 mg

Product Summary

What Is Aspadol?

Aspadol 100 mg tablet is a Tapentadol brand drug that is prescribed for treating both acute and chronic pain. Tapentadol is an opioid pain medication prescribed for the treatment of moderate to severe body pain.

With a dual mechanism of action, its use was approved by the FDA in 2008.

Formulation And List Of Ingridients

Aspadol is available in two formulations- Immediate-Release tablets and Extended-release tablets.

• An immediate-release tablet dissolves and releases its active ingredient quickly after you take it. Thus, they start working right away.
• On the other hand, an extended-release tablet is designed to dissolve slowly over time, gradually releasing its active ingredient. The extended-release tablet of Aspadol is also available in higher dosage strength, which is Aspadol ER 200 mg

Formulation: In addition to Tapentadol, the active compound, it also contains a few inactive compounds, including Microcrystalline Cellulose, Povidone K 30 USP, Magnesium Stearate, Colloidal Silicon Dioxide, and Croscarmellose sodium.

Aspadol 100mg Uses

Aspadol is prescribed to relieve acute pain resulting from surgery, back pain, or injury. It is also used for chronic pain conditions when other pain relievers are ineffective, such as diabetic neuropathy, post-operative pain, and fibromyalgia.

Benefits Of Aspadol Tablets

The three key benefits of Aspadol that make it a better choice of pain medication are listed below.

• Aspadol has a better safety profile with a lower risk of side effects compared to traditional opioid pain medication.
• It is one of the most affordable Tapentadol brand drugs available in the market.
• The action of Aspadol 100 mg (IR) lasts for 4 to 6 hours, whereas the Extended-Release (ER) tablets work for 12 hours.

How Does Aspadol 100mg Work?

Tapentadol, the active ingredient in Aspadol, has a dual mode of action-

• Mu-opioid receptor agonist- It activates the opioid receptors in the central nervous system, which helps reduce the perception of pain.
• Norepinephrine reuptake inhibitor (NRI)- It inhibits the reuptake of norepinephrine, a neurotransmitter involved in pain relief. This increases its levels and contributes to pain relief.

The action of Aspadol 100 mg begins within 30 minutes of intake, and its action lasts for about 4 to 6 hours.

Dosage Guidelines

The Aspadol 100 mg tablets can be taken two to three times daily. The maximum daily dosage of Aspadol is 600 mg.

No change in the dosage should be done without consulting a doctor.

Missed Dose

Take the missed dose as soon as you remember. If it is already time for your next dose, skip the missed dose and continue with your regular dosing schedule.

Alternative Dose

Beginners can start with a lower dose, such as Topcynta 50 mg. The dosage strength can be gradually increased based on the severity of the pain. Such people can take Tapaday 200 mg two to three daily.

For other brand drugs of Tapentadol with the same dosage strength, take Tapaday 100 mg, or Tap 100 mg.

Direction Of Use

• Swallow Aspasol 100 mg with water without breaking or crushing it.
• It can be taken with or without a meal.
• Take the medicine at a fixed time for better results.
• Do not abruptly discontinue the intake of Aspadol, as it can result in withdrawal symptoms. Consult a doctor before discontinuing Aspadol 100 tablets.

Side Effects Of Aspadol Tab 100mg

The common side effects of Tapentadol include-

• Dizziness
• Lightheadedness
• Drowsiness
• Nausea
• Dry Mouth
• Vomiting

Serious side effects may include respiratory depression, severe hypotension, and addiction or dependence with long-term use. The other side effects that must be reported to a doctor immediately include-

• Itching
• Difficulty breathing or swallowing
• Feeling overheated
• Hives
• Feeling lightheaded
• Agitation
• Hallucinations

Precaution And Warnings

Alcohol

Avoid taking Aspadol with alcohol to prevent dizziness and drowsiness.

Pregnancy

Aspadol 100 tablets is a category C medication and are not advisable during pregnancy as it can affect the developing baby.

Driving

Aspadol tablets can cause dizziness and drowsiness, making it unsafe to drive or use heavy machinery.

Breastfeeding

It is unsafe to breastfeed while taking Aspadol as it can pass into the mother’s milk to affect the growth and development of the baby. Do not feed the baby for 3 to 4 hours of taking Aspadol 100 mg.

Kidney

People with kidney disorders are advised to take Aspadol after consulting a doctor. Such patients may also require dosage adjustment.

Liver

Take Aspadol 100 mg tablets with caution if you have a liver disorder, as it may affect the metabolic activity of the medication.

Fertility

Aspadol 100mg tablets can decrease fertility in men and women. Consult a doctor before taking the medication.

Storage And Disposal

Store the Aspadol 100 mg tablets at room temperature, away from excess moisture and heat. Dispose of any medication that is not needed or expired by flushing them down the toilet.

Drug Interaction Of Aspadol 100 mg

Aspadol 100 tablets, when taken with other medications and supplements, can result in drug interaction, lowering its effectiveness and increasing the risk of side effects.

Medications that are not advised to be taken with Aspadol and can result in severe to moderate interaction are listed in the table below.

In addition to the medication listed here, always consult a doctor before taking any medication with Aspadol 100 mg.